Paul Awolade
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Explore the profile of Paul Awolade including associated specialties, affiliations and a list of published articles.
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23
Citations
216
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Recent Articles
11.
Kumar V, Dhawan S, Girase P, Awolade P, Shinde S, Karpoormath R, et al.
Curr Med Chem
. 2021 Mar;
28(33):6805-6845.
PMID: 33749549
Chalcones are an interesting class of compounds endowed with a plethora of biological activities beneficial to human health. These chemotypes have continued to attract increased research attention over the years;...
12.
Seboletswe P, Awolade P, Singh P
ChemMedChem
. 2021 Mar;
16(13):2050-2067.
PMID: 33724717
Heterocyclic compounds constitute a unique class of organic compounds endowed with a wide range of synthetic and pharmaceutical applications. Pyrimidinones and their fused analogues have received focused attention in this...
13.
Shalini , Kumar S, Gendrot M, Fonta I, Mosnier J, Cele N, et al.
ACS Med Chem Lett
. 2020 Dec;
11(12):2544-2552.
PMID: 33335678
A series of amide tethered 4-aminoquinoline-naphthalimide hybrids has been synthesized to assess their in vitro antiplasmodial potential against chloroquine-susceptible (3D7) and chloroquine-resistant (W2) strains of . The most active and...
14.
Awolade P, Cele N, Ebenezer O, Kerru N, Gummidi L, Gu L, et al.
Anticancer Agents Med Chem
. 2020 Sep;
21(10):1228-1239.
PMID: 32990543
Background: The persistence of breast cancer as the leading cause of mortality among women, coupled with drug resistance to tamoxifen, the standard endocrine therapy for the disease, exacts continuous attention....
15.
Rani A, Johansen M, Roquet-Baneres F, Kremer L, Awolade P, Ebenezer O, et al.
Bioorg Med Chem Lett
. 2020 Sep;
30(22):127576.
PMID: 32980514
A series of 4-aminoquinoline-isoindoline-dione-isoniazid triads were synthesized and assessed for their anti-mycobacterial activities and cytotoxicity. Most of the synthesized compounds exhibited promising activities against the mc6230 strain of M. tuberculosis...
16.
Gummidi L, Kerru N, Awolade P, Raza A, Sharma A, Singh P
Bioorg Med Chem Lett
. 2020 Sep;
30(22):127544.
PMID: 32920143
New indole-tethered [1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one (8a-j) and [1,3,4]oxadiazolo[3,2-a]pyrimidin-5-one hybrids (9a-e) were synthesized using [4+2] cycloaddition reactions of functionalized 1,3-diazabuta-1,3-dienes with indole-ketenes. All molecular hybrids were structurally characterized by spectroscopic techniques (IR, NMR,...
17.
Awolade P, Cele N, Kerru N, Singh P
Mol Divers
. 2020 Jun;
25(4):2201-2218.
PMID: 32507981
Antimicrobial resistance has become a significant threat to global public health, thus precipitating an exigent need for new drugs with improved therapeutic efficacy. In this regard, molecular hybridization is deemed...
18.
Awolade P, Cele N, Kerru N, Gummidi L, Oluwakemi E, Singh P
Eur J Med Chem
. 2019 Dec;
187:111921.
PMID: 31835168
The emergence of disease and dearth of effective pharmacological agents on most therapeutic fronts, constitutes a major threat to global public health and man's existence. Consequently, this has created an...
19.
Rani A, Kumar S, Legac J, Adeniyi A, Awolade P, Singh P, et al.
Future Med Chem
. 2019 Dec;
12(3):193-205.
PMID: 31802710
WHO Malaria report 2017 estimated 216 million cases of malaria and 445,000 deaths worldwide, with 91% of deaths affecting the African region. Microwave promoted the synthesis of cycloalkyl amine substituted...
20.
Synthesis, Cytotoxicity and Antimicrobial Evaluation of New Coumarin-Tagged β-Lactam Triazole Hybrid
Dhawan S, Awolade P, Kisten P, Cele N, Pillay A, Saha S, et al.
Chem Biodivers
. 2019 Dec;
17(1):e1900462.
PMID: 31788939
A series of coumarin-tagged β-lactam triazole hybrids (10a-10o) were synthesized and tested for their cytotoxic activity against MDA-MB-231 (triple negative breast cancer), MCF-7 (estrogen receptor positive breast cancer (ER+)) and...