Gabriele Giliberti
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Explore the profile of Gabriele Giliberti including associated specialties, affiliations and a list of published articles.
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27
Citations
254
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Recent Articles
1.
Sanna G, Madeddu S, Murgia G, Serreli G, Begala M, Caboni P, et al.
Viruses
. 2020 Jun;
12(6).
PMID: 32575585
Historically, natural products have been the most successful source of inspiration for the development of new drugs. Members of the Thymelaeaceae family have been of interest owing to their excellent...
2.
Sanna G, Madeddu S, Giliberti G, Piras S, Struga M, Wrzosek M, et al.
Molecules
. 2018 Oct;
23(10).
PMID: 30301264
A series of 2-(1-indol-3-yl)ethylthiourea derivatives were prepared by condensation of 2-(1-indol-3-yl)ethanamine with appropriate aryl/alkylisothiocyanates in anhydrous media. The structures of the newly synthesized compounds were confirmed by spectroscopic analysis and...
3.
Bielenica A, Sanna G, Madeddu S, Giliberti G, Stefanska J, Koziol A, et al.
Molecules
. 2018 Sep;
23(10).
PMID: 30248936
4-Chloro-3-nitrophenylthioureas ⁻ were synthesized and tested for their antimicrobial and cytotoxic activities. Compounds exhibited high to moderate antistaphylococcal activity against both standard and clinical strains (MIC values 2⁻64 μg/mL). Among...
4.
Carta A, Sanna G, Briguglio I, Madeddu S, Vitale G, Piras S, et al.
Eur J Med Chem
. 2018 Jan;
145:559-569.
PMID: 29339251
Enteroviruses are among the most common and important human pathogens for which there are no specific antiviral agents approved by the US Food and Drug Administration so far. Particularly, coxsackievirus...
5.
Bielenica A, Szulczyk D, Olejarz W, Madeddu S, Giliberti G, Materek I, et al.
Biomed Pharmacother
. 2017 Aug;
94:804-812.
PMID: 28802233
On the basis of recently reported biologically active 3-(trifluoromethyl)phenylthioureas, a series of diaryl derivatives incorporating 1H-tetrazol-5-yl (1a-11a, 1a'-11a') and 1,3-thiazolidin-4-one (1b-11b) scaffolds were synthesized. The synthesis pathway was confirmed by...
6.
Bielenica A, Sanna G, Madeddu S, Struga M, Jozwiak M, Koziol A, et al.
Chem Biol Drug Des
. 2017 Apr;
90(5):883-891.
PMID: 28434186
Thiourea derivatives have been reported to possess many biological activities, among them antiviral and antitumoral properties. As part of our continuing effort to develop new active compounds, we report the...
7.
Sanna G, Madeddu S, Giliberti G, Ntalli N, Cottiglia F, De Logu A, et al.
PLoS One
. 2015 Oct;
10(10):e0141272.
PMID: 26485025
The biological diversity of nature is the source of a wide range of bioactive molecules. The natural products, either as pure compounds or as standardized plant extracts, have been a...
8.
Briguglio I, Loddo R, Laurini E, Fermeglia M, Piras S, Corona P, et al.
Eur J Med Chem
. 2015 Oct;
105:63-79.
PMID: 26479028
Linear aromatic N-tricyclic compounds with promising antiviral activity and minimal cytotoxicity were prepared and analyzed in the last years. Specifically, the pyrido[2,3-g]quinoxalinone nucleus was found endowed with high potency against...
9.
Loddo R, Novelli F, Sparatore A, Tasso B, Tonelli M, Boido V, et al.
Bioorg Med Chem
. 2015 Oct;
23(21):7024-34.
PMID: 26443549
A library of 64 benzotriazole derivatives (17 of which were [4-(benzotriazol-2-yl)phenoxy]alkanoic acids) were screened for antiviral activity against a panel of twelve DNA and RNA viruses. Twenty-six compounds (12 of...
10.
Bielenica A, Stefanska J, Stepien K, Napiorkowska A, Augustynowicz-Kopec E, Sanna G, et al.
Eur J Med Chem
. 2015 Jun;
101:111-25.
PMID: 26119992
A total of 31 of thiourea derivatives was prepared reacting 3-(trifluoromethyl)aniline and commercial aliphatic and aromatic isothiocyanates. The yields varied from 35% to 82%. All compounds were evaluated in vitro...