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Vikas N Telvekar

Explore the profile of Vikas N Telvekar including associated specialties, affiliations and a list of published articles. Areas
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Articles 11
Citations 61
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Recent Articles
1.
Gokhale K, Telvekar V
Chem Biol Drug Des . 2020 Aug; 97(1):148-156. PMID: 32745362
Emergence of MDR-TB and XDR-TB led to the failure of available anti-tubercular drugs. In order to explore, identify and develop new anti-tubercular drugs, novel peptidomimetic series of Mtb-peptide deformylase (PDF)...
2.
Mali J, Sutar Y, Pahelkar A, Verma P, Telvekar V
Chem Biol Drug Des . 2019 Oct; 95(1):174-181. PMID: 31581353
The discovery of antibiotics around the middle twentieth century led to a decrease in the interest in antimycobacterial fatty acids. In order to re-establish the importance of naturally abundant fatty...
3.
Sutar Y, Mali J, Telvekar V, Rajmani R, Singh A
Eur J Med Chem . 2019 Sep; 183:111713. PMID: 31557610
Tuberculosis (TB) caused by Mycobacterium tuberculosis (Mtb) has become the world's leading killer disease due to a single infectious agent which survives in the host macrophage for the indefinite period....
4.
Sutar Y, Telvekar V
Mater Sci Eng C Mater Biol Appl . 2018 Sep; 92:393-406. PMID: 30184765
The effective delivery of low potency anticancer drug is a major challenge. The present study introduces the novel chitosan-polylactic acid (CS-PLA)-drug conjugate and its transferrin receptor targeted polyelectrolyte complex nanoparticles...
5.
Siddiki A, Bairwa V, Telvekar V
Comb Chem High Throughput Screen . 2014 Mar; 17(7):630-8. PMID: 24625232
A series of structurally novel, (E)-N'-(4-aryloxybenzylidene)-1H-benzimidazole-2-carbohydrazide derivatives were synthesized by molecular hybridization technique. All these compounds were evaluated against Mycobacterium tuberculosis H37Rv strains using Resazurin Microtiter assay (REMA) method. These...
6.
Patel K, Telvekar V
Eur J Med Chem . 2014 Feb; 75:43-56. PMID: 24530490
The analogs of N-[4-(piperazin-1-yl)phenyl]cinnamamide were designed and synthesized by molecular hybridization approach in which part C of the designed molecule was linked through amide and carbamate functionality that improves the...
7.
Bairwa V, Telvekar V
Comb Chem High Throughput Screen . 2012 Nov; 16(3):244-7. PMID: 23176058
Molecular hybridization approach was used to synthesize substituted 2-(2-(4-aryl oxy benzylidene) hydrazinyl)benzo thiazole derivatives with 2-hydrazinobenzothiazole and 4-(alicycli/aryl/biaryl/heteroaryl oxy)benzaldehyde as new anti-TB agents. The synthesized compounds, when tested against H37Rv...
8.
Telvekar V, Belubbi A, Bairwa V, Satardekar K
Bioorg Med Chem Lett . 2012 Feb; 22(6):2343-6. PMID: 22365752
Tuberculosis constitutes today a serious threat to human health worldwide, aggravated by the increasing number of identified multi-drug resistant strains of Mycobacterium tuberculosis (Mtb), its causative agent, as well as...
9.
Telvekar V, Bairwa V, Satardekar K, Bellubi A
Bioorg Med Chem Lett . 2011 Nov; 22(1):649-52. PMID: 22079026
A series of structurally novel, substituted 2-(2-(4-aryloxybenzylidene) hydrazinyl)benzothiazole derivatives incorporating 2-hydrazinyl benzothiazole and 4-(aryloxy)benzaldehyde were designed and synthesized using molecular hybridization approach. All the synthesized compounds exhibited promising activity (MIC...
10.
Telvekar V, Patel K
Chem Biol Drug Des . 2011 Apr; 78(1):150-60. PMID: 21518263
To elucidate the crucial structural features for the HIV-1 integrase inhibitors, a three-dimensional pharmacophore model was developed based on N-methyl pyrimidones, dihydroxypyrimidines, and bicyclic pyrimidinones derivatives using Phase. N-methyl pyrimidone...