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Ricardo Macarron

Explore the profile of Ricardo Macarron including associated specialties, affiliations and a list of published articles. Areas
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Articles 21
Citations 799
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Recent Articles
1.
Reis E, Buonpane R, Celik H, Marty C, Lei A, Jobe F, et al.
Blood . 2024 Sep; 144(22):2336-2348. PMID: 39255409
Mutations in calreticulin (mutCALR) are the second most common drivers of myeloproliferative neoplasms (MPNs) and yet, the current therapeutic landscape lacks a selective agent for mutCALR-expressing MPNs. Here, we show...
2.
Hummel J, Xiao K, Yang J, Epling L, Mukai K, Ye Q, et al.
J Med Chem . 2024 Feb; 67(4):3112-3126. PMID: 38325398
CDK2 is a critical regulator of the cell cycle. For a variety of human cancers, the dysregulation of CDK2/cyclin E1 can lead to tumor growth and proliferation. Historically, early efforts...
3.
Rapiteanu R, Karagyozova T, Zimmermann N, Singh K, Wayne G, Martufi M, et al.
Eur Respir J . 2020 Feb; 55(5). PMID: 32060058
No abstract available.
4.
Chakravorty S, Chan J, Greenwood M, Popa-Burke I, Remlinger K, Pickett S, et al.
SLAS Discov . 2018 Apr; 23(6):532-545. PMID: 29699447
High-throughput screening (HTS) hits include compounds with undesirable properties. Many filters have been described to identify such hits. Notably, pan-assay interference compounds (PAINS) has been adopted by the community as...
5.
Lu Q, Livi G, Modha S, Yusa K, Macarron R, Dow D
Expert Opin Drug Discov . 2017 Apr; 12(6):541-552. PMID: 28388235
The analysis of pharmaceutical industry data indicates that the major reason for drug candidates failing in late stage clinical development is lack of efficacy, with a high proportion of these...
6.
Powell D, Hertzberg R, Macarron R
Methods Mol Biol . 2016 Jun; 1439:1-32. PMID: 27316985
HTS remains at the core of the drug discovery process, and so it is critical to design and implement HTS assays in a comprehensive fashion involving scientists from the disciplines...
7.
Macarron R
Nat Chem Biol . 2015 Oct; 11(12):904-5. PMID: 26479440
No abstract available.
8.
Macarron R, Luengo J
Future Med Chem . 2011 Apr; 3(5):505-7. PMID: 21526891
No abstract available.
9.
Macarron R, Banks M, Bojanic D, Burns D, Cirovic D, Garyantes T, et al.
Nat Rev Drug Discov . 2011 Mar; 10(3):188-95. PMID: 21358738
High-throughput screening (HTS) has been postulated in several quarters to be a contributory factor to the decline in productivity in the pharmaceutical industry. Moreover, it has been blamed for stifling...
10.
Macarron R, Hertzberg R
Mol Biotechnol . 2010 Sep; 47(3):270-85. PMID: 20865348
High throughput screening (HTS) is at the core of the drug discovery process, and so it is critical to design and implement HTS assays in a comprehensive fashion involving scientists...