Greg Delahanty
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Explore the profile of Greg Delahanty including associated specialties, affiliations and a list of published articles.
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7
Citations
182
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Recent Articles
1.
Hin N, Alt J, Zimmermann S, Delahanty G, Ferraris D, Rojas C, et al.
Bioorg Med Chem
. 2014 Oct;
22(21):5831-7.
PMID: 25288495
A series of Arg-Phe-NH2 peptidomimetics containing an Arg mimetic were synthesized and tested as agonists of human MrgX1, rat MrgC, and mouse MrgC11 receptors. As predicted from the previously established...
2.
Ferraris D, Duvall B, Delahanty G, Mistry B, Alt J, Rojas C, et al.
J Med Chem
. 2014 Feb;
57(6):2582-8.
PMID: 24520856
Several 2'-fluorinated tetrahydrouridine derivatives were synthesized as inhibitors of cytidine deaminase (CDA). (4R)-2'-Deoxy-2',2'-difluoro-3,4,5,6-tetrahydrouridine (7a) showed enhanced acid stability over tetrahydrouridine (THU) 5 at its N-glycosyl bond. As a result, compound...
3.
Shukla K, Ferraris D, Thomas A, Stathis M, Duvall B, Delahanty G, et al.
J Med Chem
. 2012 Nov;
55(23):10551-63.
PMID: 23151085
Bis-2-(5-phenylacetamido-1,2,4-thiadiazol-2-yl)ethyl sulfide (BPTES) is a potent and selective allosteric inhibitor of kidney-type glutaminase (GLS) that has served as a molecular probe to determine the therapeutic potential of GLS inhibition. In...
4.
Stoermer D, Vitharana D, Hin N, Delahanty G, Duvall B, Ferraris D, et al.
J Med Chem
. 2012 May;
55(12):5922-32.
PMID: 22642259
A series of thiol-based glutamate carboxypeptidase II (GCPII) inhibitors have been synthesized with either a 3-(mercaptomethyl)benzoic acid or 2-(2-mercaptoethyl)benzoic acid scaffold. Potent inhibitors were identified from each of the two...
5.
Grella B, Adams J, Berry J, Delahanty G, Ferraris D, Majer P, et al.
Bioorg Med Chem Lett
. 2010 Nov;
20(24):7222-5.
PMID: 21074428
A series of N-substituted 3-(2-mercaptoethyl)-1H-indole-2-carboxylic acids were synthesized as inhibitors of glutamate carboxypeptidase II (GCPII). Those containing carboxybenzyl or carboxyphenyl groups at the N-position exhibited potent inhibitory activity against GCPII....
6.
Majer P, Hin B, Stoermer D, Adams J, Xu W, Duvall B, et al.
J Med Chem
. 2006 May;
49(10):2876-85.
PMID: 16686531
A series of thiol-based inhibitors containing a benzyl moiety at the P1' position have been synthesized and tested for their abilities to inhibit glutamate carboxypeptidase II (GCP II). 3-(2-Carboxy-5-mercaptopentyl)benzoic acid...
7.
Majer P, Jackson P, Delahanty G, Grella B, Ko Y, Li W, et al.
J Med Chem
. 2003 May;
46(10):1989-96.
PMID: 12723961
A series of 2-(thioalkyl)pentanedioic acids were synthesized and evaluated as inhibitors of glutamate carboxypeptidase II (GCP II, EC 3.4.17.21). The inhibitory potency of these thiol-based compounds against GCP II was...