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Kartik Keertikar

Explore the profile of Kartik Keertikar including associated specialties, affiliations and a list of published articles. Areas
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Citations 31
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Recent Articles
1.
Bungard C, Williams P, Schulz J, Wiscount C, Holloway M, Loughran H, et al.
ACS Med Chem Lett . 2017 Dec; 8(12):1292-1297. PMID: 29259750
Using the HIV-1 protease binding mode of and as inspiration, a novel aspartate binding bicyclic piperazine sulfonamide core was designed and synthesized. The resulting HIV-1 protease inhibitor containing this core...
2.
Dwyer M, Keertikar K, Paruch K, Alvarez C, Labroli M, Poker C, et al.
Bioorg Med Chem Lett . 2013 Oct; 23(22):6178-82. PMID: 24091081
The synthesis and hit-to-lead SAR development from a pyrazolo[1,5-a]pyrimidine-derived hit 5 to the identification of a series of potent, pan-Pim inhibitors such as 11j are described.
3.
Labroli M, Paruch K, Dwyer M, Alvarez C, Keertikar K, Poker C, et al.
Bioorg Med Chem Lett . 2010 Nov; 21(1):471-4. PMID: 21094607
Previous efforts by our group have established pyrazolo[1,5-a]pyrimidine as a viable core for the development of potent and selective CDK inhibitors. As part of an effort to utilize the pyrazolo[1,5-a]pyrimidine...