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Jason Laskey

Explore the profile of Jason Laskey including associated specialties, affiliations and a list of published articles. Areas
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Articles 8
Citations 380
Followers 0
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Recent Articles
1.
Chang W, Altman M, Lesburg C, Perera S, Piesvaux J, Schroeder G, et al.
J Med Chem . 2022 Mar; 65(7):5675-5689. PMID: 35332774
Stereochemically and structurally complex cyclic dinucleotide-based stimulator of interferon genes (STING) agonists were designed and synthesized to access a previously unexplored chemical space. The assessment of biochemical affinity and cellular...
2.
Perera S, Kopinja J, Ma Y, Muise E, Laskey J, Chakravarthy K, et al.
Mol Cancer Ther . 2021 Nov; 21(2):282-293. PMID: 34815361
The innate immune agonist STING (STimulator of INterferon Genes) binds its natural ligand 2'3'-cGAMP (cyclic guanosine-adenosine monophosphate) and initiates type I IFN production. This promotes systemic antigen-specific CD8 T-cell priming...
3.
Wang Y, Zhang K, Georgiev P, Wells S, Xu H, Lacey B, et al.
PLoS One . 2020 Dec; 15(12):e0243145. PMID: 33270695
Hematopoietic progenitor kinase 1 (HPK1), a hematopoietic cell-specific Ste20-related serine/threonine kinase, is a negative regulator of signal transduction in immune cells, including T cells, B cells, and dendritic cells (DCs)....
4.
Lacey B, Xu Z, Chai X, Laskey J, Fradera X, Mittal P, et al.
SLAS Discov . 2020 Aug; 26(1):88-99. PMID: 32844715
Hematopoietic progenitor kinase 1 (HPK1), also referred to as mitogen-activated protein kinase kinase kinase kinase 1 (MAP4K1), is a serine/threonine kinase that negatively regulates T-cell signaling by phosphorylating Ser376 of...
5.
Pan B, Perera S, Piesvaux J, Presland J, Schroeder G, Cumming J, et al.
Science . 2020 Aug; 369(6506). PMID: 32820094
Pharmacological activation of the STING (stimulator of interferon genes)-controlled innate immune pathway is a promising therapeutic strategy for cancer. Here we report the identification of MSA-2, an orally available non-nucleotide...
6.
McLeod R, Angagaw M, Baral T, Liu L, Moniz R, Laskey J, et al.
Oncotarget . 2018 Oct; 9(77):34459-34470. PMID: 30349641
Carcinoembryonic antigen-related cell adhesion molecule 1 (CEACAM1) has been reported to mediate both tumorigenic and anti-tumor effects . Blockade of the CEACAM1 signaling pathway has recently been implicated as a...
7.
Stoeck A, Lejnine S, Truong A, Pan L, Wang H, Zang C, et al.
Cancer Discov . 2014 Aug; 4(10):1154-67. PMID: 25104330
Unlabelled: Next-generation sequencing was used to identify Notch mutations in a large collection of diverse solid tumors. NOTCH1 and NOTCH2 rearrangements leading to constitutive receptor activation were confined to triple-negative...
8.
Zhang W, Zhu J, Efferson C, Ware C, Tammam J, Angagaw M, et al.
Cancer Res . 2009 Sep; 69(18):7466-72. PMID: 19738074
Androgen receptors have been shown to play a critical role in prostate cancer. We used ultrasound imaging techniques to track tumor response to antiandrogen and rapamycin treatment in a prostate-specific...