Carmela Inglese
Overview
Explore the profile of Carmela Inglese including associated specialties, affiliations and a list of published articles.
Author names and details appear as published. Due to indexing inconsistencies, multiple individuals may share a name, and a single author may have variations. MedLuna displays this data as publicly available, without modification or verification
Snapshot
Snapshot
Articles
16
Citations
143
Followers
0
Related Specialties
Related Specialties
Top 10 Co-Authors
Top 10 Co-Authors
Published In
Affiliations
Affiliations
Soon will be listed here.
Recent Articles
1.
Munro T, Huang X, Inglese C, Perrone M, Vant Veer A, Carroll F, et al.
PLoS One
. 2013 Aug;
8(8):e70701.
PMID: 23976952
Background: Nor-BNI, GNTI and JDTic induce selective κ opioid antagonism that is delayed and extremely prolonged, but some other effects are of rapid onset and brief duration. The transient effects...
2.
Perrone M, Inglese C, Berardi F, Leopoldo M, Perrone R, Colabufo N
J Pharmacol Toxicol Methods
. 2012 Dec;
67(1):5-8.
PMID: 23234641
Introduction: P-glycoprotein (P-gp) plays a crucial role in beta-amyloid efflux from the blood-brain barrier thus becoming a promising pharmacological target in the treatment of Alzheimer's disease (AD). The increase of...
3.
Contino M, Cantore M, Capparelli E, Perrone M, Niso M, Inglese C, et al.
ChemMedChem
. 2012 Jan;
7(3):391-5.
PMID: 22213697
No abstract available.
4.
Inglese C, Perrone M, Berardi F, Perrone R, Colabufo N
Curr Drug Metab
. 2011 Mar;
12(8):702-12.
PMID: 21434860
P-glycoprotein (P-gp) is involved in MDR and in neurodegenerative disorders such as Parkinson disease (PD), Alzheimer disease (AD) and epilepsy. Cytochrome P450 enzymes (CYP450s) catalyze the metabolism of a wide...
5.
Colabufo N, Berardi F, Perrone M, Capparelli E, Cantore M, Inglese C, et al.
Curr Top Med Chem
. 2010 Jul;
10(17):1703-14.
PMID: 20645922
In recent years, several PET tracers for monitoring the activity and expression of P-gp at the BBB have been tested. P-gp substrates such as [(11)C]verapamil and [(11)C]loperamide can be employed...
6.
Colabufo N, Contino M, Inglese C, Niso M, Perrone R, Roperto S, et al.
Cent Nerv Syst Agents Med Chem
. 2009 Dec;
9(3):161-71.
PMID: 20021350
Methods for addressing sigma receptor affinity and activity have been explored and although several protocols have been employed, only few procedures resulted reliable. Sigma-1 receptor affinity protocol using guinea-pig brain...
7.
Colabufo N, Berardi F, Cantore M, Contino M, Inglese C, Niso M, et al.
J Med Chem
. 2009 Nov;
53(5):1883-97.
PMID: 19924994
No abstract available.
8.
Lacivita E, Leopoldo M, Masotti A, Inglese C, Berardi F, Perrone R, et al.
J Med Chem
. 2009 Aug;
52(23):7892-6.
PMID: 19705871
A series of "long-chain" 1-(2-methoxyphenyl)piperazine derivatives containing an environment-sensitive fluorescent moiety (4-amino-1,8-naphthalimide, 4-dimethylaminophthalimide, dansyl) was synthesized. The compounds displayed very high to moderate 5-HT(1A) receptor affinity and good fluorescence properties....
9.
Colabufo N, Berardi F, Perrone M, Cantore M, Contino M, Inglese C, et al.
ChemMedChem
. 2009 Jan;
4(2):188-95.
PMID: 19140144
2-Aryloxazole and 2-arylthiazole derivatives were evaluated for their inhibitory activity toward P-glycoprotein (P-gp) as well as their selectivity toward other ABC transporters involved in multi-drug resistance such as BCRP and...
10.
Colabufo N, Pagliarulo V, Berardi F, Contino M, Inglese C, Niso M, et al.
Eur J Pharmacol
. 2008 Nov;
601(1-3):38-42.
PMID: 18992739
Prolonged bicalutamide treatment induced pathology regression although relapses with a more aggressive form of prostate cancer have been observed. This failure could be due to androgen receptor mutation. In the...