S A Yarkov
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Explore the profile of S A Yarkov including associated specialties, affiliations and a list of published articles.
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4
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12
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Recent Articles
1.
[PHARMACOLOGICAL STUDY OF NEW COMPOUNDS ACTING AS REGULATORS OF 18-KDA TRANSLOCATOR PROTEIN LIGANDS]
Yarkov S, Mokrov G, Gudasheva T, Yarkova M, Seredenin S
Eksp Klin Farmakol
. 2016 May;
79(1):7-11.
PMID: 27159950
The interaction of new original 1-arylpyrrolo[1,2-a]pyrazine-3-carboxamide derivatives with mitochondrial translocator protein (MTP) 18 kDa has been studied by radioligand binding assay. Compounds GML-1 (Ki = 5.2 x 10⁻⁸ M) and...
2.
Gudasheva T, Deeva O, Mokrov G, Yarkov S, Yarkova M, Seredenin S
Dokl Biochem Biophys
. 2015 Nov;
464:290-3.
PMID: 26518550
On the basis of the structure of Alpidem, a pyrazolopyrimidine ligand of the translocator protein (TSPO), a dipeptide TSPO ligand, N-carbobenzoxy-L-tryptophanyl-L-isoleucine amide (GD-23), was designed and synthesized using our own...
3.
Povarnina P, Yarkov S, Gudasheva T, Yarkova M, Seredenin S
Acta Naturae
. 2015 Oct;
7(3):108-12.
PMID: 26483966
The translocator protein (TSPO) promotes the translocation of cholesterol to the inner mitochondrial membrane and mediates steroid formation. In this study, we first report on a biological evaluation of the...
4.
Mokrov G, Deeva O, Gudasheva T, Yarkov S, Yarkova M, Seredenin S
Bioorg Med Chem
. 2015 May;
23(13):3368-78.
PMID: 25937237
A series of 1-arylpyrrolo[1,2-a]pyrazine-3-carboxamides were designed and synthesized as 18kDa translocator protein (TSPO) ligands. Anxiolytic-like activity of compounds was evaluated in the open field test and elevated plus maze test....