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» Authors » Bandar E Aldhubiab

Bandar E Aldhubiab

Explore the profile of Bandar E Aldhubiab including associated specialties, affiliations and a list of published articles. Areas
Snapshot
Articles 22
Citations 160
Followers 0
Related Specialties
Pharmacology
Biology
Biochemistry
Top 10 Co-Authors
Katharigatta N Venugopala
Mahesh Attimarad
Anroop B Nair
Sandeep Chandrashekharappa
Mohamed A Morsy
Nagaraja Sreeharsha
Melendhran Pillay
Deepak Chopra
Rashmi Venugopala
Bharti Odhav
Published In
Molecules
Antibiotics (Basel)
Drug Des Devel Ther
J Biomol Struct Dyn
J Microencapsul
Affiliations
Soon will be listed here.
Recent Articles
1.
Identification of potent indolizine derivatives against Mycobacterial tuberculosis: In vitro anti-TB properties, in silico target validation, molecular docking and dynamics studies
Venugopala K, Chandrashekharappa S, Deb P, Al-Shari N, Pillay M, Tiwari P, et al.
Int J Biol Macromol . 2024 Jun; 274(Pt 2):133285. PMID: 38925196
In the current study, two sets of compounds: (E)-1-(2-(4-substitutedphenyl)-2-oxoethyl)-4-((hydroxyimino)methyl)pyridinium derivatives (3a-3e); and (E)-3-(substitutedbenzoyl)-7-((hydroxyimino)methyl)-2-substitutedindolizine-1-carboxylate derivatives (5a-5j), were synthesized and biologically evaluated against two strains of Mycobacterial tuberculosis (ATCC 25177) and multi-drug...
2.
Computational Design, Synthesis, and Pharmacological Evaluation of Naproxen-Guaiacol Chimera for Gastro-Sparing Anti-Inflammatory Response by Selective COX2 Inhibition
Shinu P, Sharma M, Gupta G, Mujwar S, Kandeel M, Kumar M, et al.
Molecules . 2022 Oct; 27(20). PMID: 36296501
The 4-allyl guaiacol is a natural phenolic molecule that has been widely studied for its antioxidant capacity against reactive-oxygen-species-mediated cellular damage. Therefore, we hypothesized that concomitant use of an antioxidant...
3.
Development of Novel Unfolding Film System of Itopride Hydrochloride Using Box-Behnken Design-A Gastro Retentive Approach
Alaithan S, Raghavendra Naveen N, Goudanavar P, Bhavani P, Ramesh B, Koppuravuri N, et al.
Pharmaceuticals (Basel) . 2022 Aug; 15(8). PMID: 36015129
Currently, gastro-retentive dosage forms achieved a remarkable position among the oral drug delivery systems. This is a broadly used technique to hold the drug delivery systems for a long duration...
4.
Evaluation of the Potential of National Sharing of a Unified Progress Test Among Colleges of Pharmacy in the Kingdom of Saudi Arabia
Albekairy A, Obaidat A, Alsharidah M, Alqasomi A, Alsayari A, Albarraq A, et al.
Adv Med Educ Pract . 2021 Dec; 12:1465-1475. PMID: 34938140
Background: With the expansion in pharmacy education in Saudi Arabia, there is a pressing need to maintain quality assurance in pharmacy programs using several tools. The progress test is a...
5.
Design, Synthesis, and In Vitro Evaluation of Novel Indolyl DiHydropyrazole Derivatives as Potential Anticancer Agents
Venugopala K, Habeebuddin M, Aldhubiab B, Haq Asif A
Molecules . 2021 Sep; 26(17). PMID: 34500672
Indoles derived from both natural sources or artificial synthetic methods have been known to interact with aryl hydrocarbon receptors (AhR), and exhibit anticancer activity. In light of these attractive properties,...
6.
Anti-tubercular activity and molecular docking studies of indolizine derivatives targeting mycobacterial InhA enzyme
Venugopala K, Chandrashekharappa S, Deb P, Tratrat C, Pillay M, Chopra D, et al.
J Enzyme Inhib Med Chem . 2021 Jul; 36(1):1472-1487. PMID: 34210233
A series of 1,2,3-trisubstituted indolizines (, and ) were screened for whole-cell anti-tubercular activity against the susceptible H37Rv and multidrug-resistant (MDR) (MTB) strains. Compounds , , and were active against...
7.
Crystallography, Molecular Modeling, and COX-2 Inhibition Studies on Indolizine Derivatives
Venugopala K, Chandrashekharappa S, Tratrat C, Deb P, Nagdeve R, Nayak S, et al.
Molecules . 2021 Jul; 26(12). PMID: 34200764
The cyclooxygenase-2 (COX-2) enzyme is an important target for drug discovery and development of novel anti-inflammatory agents. Selective COX-2 inhibitors have the advantage of reduced side-effects, which result from COX-1...
8.
4-Aryl-1,4-Dihydropyridines as Potential Enoyl-Acyl Carrier Protein Reductase Inhibitors: Antitubercular Activity and Molecular Docking Study
Venugopala K, Deb P, Pillay M, Chopra D, Chandrashekharappa S, Morsy M, et al.
Curr Top Med Chem . 2020 Nov; 21(4):295-306. PMID: 33138763
Background: Tuberculosis remains one of the most deadly infectious diseases worldwide due to the emergence of multi-drug resistance (MDR) and extensively drug resistance (XDR) strains of Mycobacterium tuberculosis (MTB). Aims:...
9.
Crystallography, in Silico Studies, and In Vitro Antifungal Studies of 2,4,5 Trisubstituted 1,2,3-Triazole Analogues
Venugopala K, Khedr M, Girish Y, Bhandary S, Chopra D, Morsy M, et al.
Antibiotics (Basel) . 2020 Jun; 9(6). PMID: 32575727
A series of 2,4,5 trisubstituted-1,2,3-triazole analogues have been screened for their antifungal activity against five fungal strains, , , , , and , via a 3-[4,5-dimethylthiazol-2-yl]-2,5-diphenyltetrazolium bromide (MTT) microdilution assay....
10.
Cytotoxicity and Antimycobacterial Properties of Pyrrolo[1,2-]quinoline Derivatives: Molecular Target Identification and Molecular Docking Studies
Venugopala K, Uppar V, Chandrashekharappa S, Abdallah H, Pillay M, Deb P, et al.
Antibiotics (Basel) . 2020 May; 9(5). PMID: 32392709
A series of ethyl 1-(substituted benzoyl)-5-methylpyrrolo[1,2-]quinoline-3-carboxylates - and dimethyl 1-(substituted benzoyl)-5-methylpyrrolo[1,2-]quinoline-2,3-dicarboxylates - have been synthesized and evaluated for their anti-tubercular (TB) activities against H37Rv (American Type Culture Collection (ATCC) strain...