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Btk Inhibition: the Importance of Being Selective

Overview
Journal Blood Adv
Specialty Hematology
Date 2024 Oct 25
PMID 39453633
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References
1.
Thomas J, Sideras P, Smith C, Vorechovsky I, Chapman V, Paul W . Colocalization of X-linked agammaglobulinemia and X-linked immunodeficiency genes. Science. 1993; 261(5119):355-8. DOI: 10.1126/science.8332900. View

2.
Wang M, Rule S, Martin P, Goy A, Auer R, Kahl B . Targeting BTK with ibrutinib in relapsed or refractory mantle-cell lymphoma. N Engl J Med. 2013; 369(6):507-16. PMC: 4513941. DOI: 10.1056/NEJMoa1306220. View

3.
Kuter D, Efraim M, Mayer J, Trneny M, McDonald V, Bird R . Rilzabrutinib, an Oral BTK Inhibitor, in Immune Thrombocytopenia. N Engl J Med. 2022; 386(15):1421-1431. DOI: 10.1056/NEJMoa2110297. View

4.
Rayes J, Watson S, Nieswandt B . Functional significance of the platelet immune receptors GPVI and CLEC-2. J Clin Invest. 2019; 129(1):12-23. PMC: 6307936. DOI: 10.1172/JCI122955. View

5.
Bye A, Unsworth A, Desborough M, Hildyard C, Appleby N, Bruce D . Severe platelet dysfunction in NHL patients receiving ibrutinib is absent in patients receiving acalabrutinib. Blood Adv. 2018; 1(26):2610-2623. PMC: 5728643. DOI: 10.1182/bloodadvances.2017011999. View