A Comparison of the Influence of N-isopropyl and N-tert Butyl Substituents on the Affinity of Ligands for Sinoatrial Beta-adrenoceptors in Rat Atria and Beta-adrenoceptors Coupled to the Adenylyl Cyclase in Kitten Ventricle

Overview

Journal Naunyn Schmiedebergs Arch Pharmacol

Specialty Pharmacology

Date 1979 May 28

PMID 39258

Citations 11

Authors

A J Kaumann

T H Morris

L Birnbaumer

Affiliations

Soon will be listed here.

Citing Articles

Differences between the third cardiac beta-adrenoceptor and the colonic beta 3-adrenoceptor in the rat.

Kaumann A, Molenaar P Br J Pharmacol. 1996; 118(8):2085-98.

PMID: 8864547 PMC: 1909870. DOI: 10.1111/j.1476-5381.1996.tb15648.x.

Expression of beta 3-adrenoceptor mRNA in rat tissues.

Evans B, Papaioannou M, Bonazzi V, Summers R Br J Pharmacol. 1996; 117(1):210-6.

PMID: 8825365 PMC: 1909365. DOI: 10.1111/j.1476-5381.1996.tb15176.x.

Competitive and non-competitive interactions between specific ligands and beta-adrenoceptors in living cardiac cells.

Porzig H, Becker C, Reuter H Naunyn Schmiedebergs Arch Pharmacol. 1982; 321(2):89-99.

PMID: 6296703 DOI: 10.1007/BF00518474.

A novel analysis of concentration-dependence of partial agonism Ring-demethylation of bupranolol results in a high affinity partial agonist (K 105) for myocardial and tracheal beta-adrenoceptors.

Lemoine H, Kaumann A Naunyn Schmiedebergs Arch Pharmacol. 1982; 320(2):130-44.

PMID: 6289139 DOI: 10.1007/BF00506313.

An initial characterization of human heart beta-adrenoceptors and their mediation of the positive inotropic effects of catecholamines.

Kaumann A, Lemoine H, Morris T, Schwederski U Naunyn Schmiedebergs Arch Pharmacol. 1982; 319(3):216-21.

PMID: 6287309 DOI: 10.1007/BF00495868.

References

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Morris T, Birnbaumer L, Kaumann A . High affinity of carozolol for beta-adrenoceptors coupled to the adenylyl cyclase in ventricular myocardium of kitten and Xenopus laevis. Naunyn Schmiedebergs Arch Pharmacol. 1978; 303(3):295-7. DOI: 10.1007/BF00498057. View

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