A Convergent, Enantioselective Total Synthesis of Hapalosin: A Drug with Multidrug-Resistance Reversing Activity

Overview

Journal Angew Chem Int Ed Engl

Specialty Chemistry

Date 2018 Oct 23

PMID 30344446

Citations 6

Authors

Arun K Ghosh

Wenming Liu

Yibo Xu

Zhidong Chen

Affiliations

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Citing Articles

Synthesis of Bioactive Natural Products by Asymmetric - and -Aldol Reactions.

Ghosh A, Dawson Z Synthesis (Stuttg). 2018; 2009(17):2992-3002.

PMID: 30443084 PMC: 6233898. DOI: 10.1055/s-0029-1216941.

-1-Aminoindan-2-ol in Asymmetric Syntheses.

Ghosh A, Fidanze S, Senanayake C Synthesis (Stuttg). 2018; 1998(7):937-961.

PMID: 30393403 PMC: 6214626. DOI: 10.1055/s-1998-2092.

A Convenient Enzymatic Route to Optically Active l-Aminoindan-2-ol: Versatile Ligands for HIV-1 Protease Inhibitors and Asymmetric Syntheses.

Ghosh A, Kincaid J, Haske M Synthesis (Stuttg). 2018; 1997(5):541-544.

PMID: 30393402 PMC: 6214614. DOI: 10.1055/s-1997-1235.

Asymmetric alkylations and aldol reactions: (1,2)-2-aminocyclopentan-1-ol derived new chiral auxiliary.

Ghosh A, Cho H, Onishi M Tetrahedron Asymmetry. 2018; 8(6):821-824.

PMID: 30387787 PMC: 6207082. DOI: 10.1016/S0957-4166(97)00065-7.

Capturing the essence of organic synthesis: from bioactive natural products to designed molecules in today's medicine.

Ghosh A J Org Chem. 2010; 75(23):7967-89.

PMID: 20936876 PMC: 2993809. DOI: 10.1021/jo101606g.

References

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