Solid-phase Preparation of Amides Using N-acylbenzotriazoles

Overview

Journal Bioorg Med Chem Lett

Specialty Biochemistry

Date 2002 Jun 28

PMID 12086822

Citations 1

Authors

Alan R Katritzky

Boris V Rogovoy

Nataliya Kirichenko

Vladimir Vvedensky

Affiliations

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Abstract

Wang resin linked amines were efficiently converted into amides using acylbenzotriazoles. Cleavage of resins gave the desired amides 7Aa-Gf in 30-99% yields with good to excellent purities.

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