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A N Jain

Explore the profile of A N Jain including associated specialties, affiliations and a list of published articles. Areas
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Articles 15
Citations 740
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Recent Articles
1.
Snijders A, Nowak N, Segraves R, Blackwood S, Brown N, Conroy J, et al.
Nat Genet . 2001 Nov; 29(3):263-4. PMID: 11687795
We have assembled arrays of approximately 2,400 BAC clones for measurement of DNA copy number across the human genome. The arrays provide precise measurement (s.d. of log2 ratios=0.05-0.10) in cell...
2.
Jain A, Chin K, Borresen-Dale A, Erikstein B, Eynstein Lonning P, Kaaresen R, et al.
Proc Natl Acad Sci U S A . 2001 Jul; 98(14):7952-7. PMID: 11438741
We present a general method for rigorously identifying correlations between variations in large-scale molecular profiles and outcomes and apply it to chromosomal comparative genomic hybridization data from a set of...
3.
Jain A
J Comput Aided Mol Des . 2000 Mar; 14(2):199-213. PMID: 10721506
Recognition of small molecules by proteins depends on three-dimensional molecular surface complementarity. However, the dominant techniques for analyzing the similarity of small molecules are based on two-dimensional chemical structure, with...
4.
Ghuloum A, Sage C, Jain A
J Med Chem . 1999 May; 42(10):1739-48. PMID: 10346926
We define a novel numerical molecular representation, called the molecular hashkey, that captures sufficient information about a molecule to predict pharmaceutically interesting properties directly from three-dimensional molecular structure. The molecular...
5.
Mount J, Ruppert J, Welch W, Jain A
J Med Chem . 1999 Jan; 42(1):60-6. PMID: 9888833
IcePick is a system for computationally selecting diverse sets of molecules. It computes the dissimilarity of the surface-accessible features of two molecules, taking into account conformational flexibility. Then, the intrinsic...
6.
Ruppert J, Welch W, Jain A
Protein Sci . 1997 Mar; 6(3):524-33. PMID: 9070435
Molecular docking is a popular way to screen for novel drug compounds. The method involves aligning small molecules to a protein structure and estimating their binding affinity. To do this...
7.
Jain A
J Comput Aided Mol Des . 1996 Oct; 10(5):427-40. PMID: 8951652
Exploitation of protein structures for potential drug leads by molecular docking is critically dependent on methods for scoring putative protein-ligand interactions. An ideal function for scoring must exhibit predictive accuracy...
8.
Welch W, Ruppert J, Jain A
Chem Biol . 1996 Jun; 3(6):449-62. PMID: 8807875
Background: Molecular docking seeks to predict the geometry and affinity of the binding of a small molecule to a given protein of known structure. Rigid docking has long been used...
9.
Jain A, Harris N, Park J
J Med Chem . 1995 Apr; 38(8):1295-308. PMID: 7731016
We present enhancements to the Compass algorithm that automatically deduce interchemotype relationships and generate predictive quantitative models of receptor binding based solely on structure-activity data. We applied the technique to...
10.
Jain A, Dietterich T, Lathrop R, Chapman D, Critchlow Jr R, Bauer B, et al.
J Comput Aided Mol Des . 1994 Dec; 8(6):635-52. PMID: 7738601
Building predictive models for iterative drug design in the absence of a known target protein structure is an important challenge. We present a novel technique, Compass, that removes a major...