Structural Requirements of Imidazole Compounds to Be Inhibitors or Activators of Histamine Methyltransferase: Investigation of Histamine Analogues and H2-receptor Antagonists

Overview

Journal Agents Actions

Specialty Pharmacology

Date 1978 Jun 1

PMID 28646

Citations 9

Authors

H Barth

W Lorenz

Affiliations

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Citing Articles

Dual role of imidazole as activator/inhibitor of sweet almond () β-glucosidase.

Caramia S, Gatius A, Dal Piaz F, Gaja D, Hochkoeppler A Biochem Biophys Rep. 2017; 10:137-144.

PMID: 28955741 PMC: 5614632. DOI: 10.1016/j.bbrep.2017.03.007.

Histamine N-methyltransferase: inhibition by monoamine oxidase inhibitors.

Scott M, Weinshilboum R Agents Actions. 1993; 40(1-2):1-10.

PMID: 8147263 DOI: 10.1007/BF01976745.

Inhibition of plant and mammalian diamine oxidase by substrate analogues.

Bieganski T, Osinska Z, Maslinski C Agents Actions. 1982; 12(1-2):41-6.

PMID: 6805264 DOI: 10.1007/BF01965104.

Gastric histamine methyltransferase: different methylation rates for enantiomers of side-chain methylated histamine analogues using a highly purified enzyme preparation.

Barth H, Schunack W, Crombach M, Lorenz W Agents Actions. 1984; 14(3-4):346-50.

PMID: 6731176 DOI: 10.1007/BF01973824.

Histamine uptake and metabolism in intact isolated parietal cells.

Albinus M, SEWING K Agents Actions. 1981; 11(3):223-7.

PMID: 6266232 DOI: 10.1007/BF01967618.

References

Barth H, Crombach M, Schunack W, Lorenz W . Evidence for a less high acceptor substrate specificity of gastric histamine methyltransferase: methylation of imidazole compounds. Biochem Pharmacol. 1980; 29(10):1399-407. DOI: 10.1016/0006-2952(80)90436-0. View

Lorenz W, Reimann H, Barth H, Kusche J, Meyer R, Doenicke A . A sensitive and specific method for the determination of histomine in human whole blood and plasma. Hoppe Seylers Z Physiol Chem. 1972; 353(6):911-20. DOI: 10.1515/bchm2.1972.353.1.911. View

Barth H, Niemeyer I, Lorenz W . Similar actions of methylated histamines and histamine receptor antagonists on gastric histamine methyltransferase. Agents Actions. 1973; 3(3):173-5. DOI: 10.1007/BF01965730. View

Black J, Duncan W, Durant C, Ganellin C, Parsons E . Definition and antagonism of histamine H 2 -receptors. Nature. 1972; 236(5347):385-90. DOI: 10.1038/236385a0. View

Black J, Durant G, EMMETT J, Ganellin C . Sulphur-methylene isosterism in the development of metiamide, a new histamine H2-receptor antagonist. Nature. 1974; 248(5443):65-7. DOI: 10.1038/248065a0. View

Durant G, Ganellin C, Parsons M . Dimaprit, (S-[3-(N,N-dimethylamino)propyl]isothiourea). A highly specific histamine H2-receptor agonist. Part 2. Structure-activity considerations. Agents Actions. 1977; 7(1):39-43. DOI: 10.1007/BF01964879. View

Barth H, Niemeyer I, Lorenz W . Studies on the mode of action of histamine H1- and H2-receptor antagonists on gastric histamine methyltransferase. Agents Actions. 1973; 3(3):138-47. DOI: 10.1007/BF01965724. View

Durant G, EMMETT J, Ganellin C, Miles P, Parsons M, Prain H . Cyanoguanidine-thiourea equivalence in the development of the histamine H2-receptor antagonist, cimetidine. J Med Chem. 1977; 20(7):901-6. DOI: 10.1021/jm00217a007. View

Snyder S, Axelrod J . Sex differences and hormonal control of histamine methyltransferase activity. Biochim Biophys Acta. 1965; 111(2):416-21. DOI: 10.1016/0304-4165(65)90051-6. View

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Barth H, Niemeyer I, Lorenz W . Speculations about the binding sites of S-adenosyl-L-homocysteine and some of its synthetic analogues to histamine methyltransferase. Agents Actions. 1974; 4(3):186-8. DOI: 10.1007/BF01970266. View

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LOWRY O, ROSEBROUGH N, FARR A, RANDALL R . Protein measurement with the Folin phenol reagent. J Biol Chem. 1951; 193(1):265-75. View

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Barth H, Lorenz W, Niemeyer I . Inhibition and activation of histamine methyltransferase by methylated histamines. Hoppe Seylers Z Physiol Chem. 1973; 354(9):1021-6. DOI: 10.1515/bchm2.1973.354.2.1021. View

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Parsons M, Owen D, Ganellin C, Durant G . Dimaprit -(S-[3-(N,N-dimethylamino)prophyl]isothiourea) - a highly specific histamine H2 -receptor agonist. Part 1. Pharmacology. Agents Actions. 1977; 7(1):31-7. DOI: 10.1007/BF01964878. View

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Taylor K, Snyder S . Histamine methyltransferase: inhibition and potentiation by antihistamines. Mol Pharmacol. 1972; 8(3):300-10. View

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Maslinski S, Schippert B, Kovar K, SEWING K . Methylation of histamine in the gastric mucosa. Digestion. 1977; 15(6):497-505. DOI: 10.1159/000198040. View